| Round | Overall | Player |
|---|---|---|
| 1 | 11th | OF Jason Bay Pit |
| 2 | 14th | DH Travis Hafner Cle |
| 3 | 35th | OF Grady Sizemore Cle |
| 4 | 38th | SP Roy Oswalt Hou |
| 5 | 59th | SP Barry Zito Oak |
| 6 | 62nd | SP Mark Buehrle ChA |
| 7 | 83rd | OF J.D. Drew LAD |
| 8 | 86th | RP Ryan Dempster ChN |
| 9 | 107th | SP Carlos Silva Min |
| 10 | 110th | RP Danys Baez Bal |
| 11 | 131st | SP Freddy Garcia ChA |
| 12 | 134th | 2B Tadahito Iguchi ChA |